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SRPIN340

SRPK inhibitor
Catalog No. S21-901


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Catalog No. Pack Size Price (USD)
S21-901-05 5 mg $83
S21-901-25 25 mg $303
S21-901-BULK BULK Contact Us  


Overview:

Serine arginine protein kinase (SRPK) 1 inhibitor (Ki = 0.89 µM)1. Inhibits SRPK2 at higher concentrations. Does not significantly inhibit other SRPKs such as CLK1 and CLK4, or other classes of SR kinases.

References:


1. T Fukuhara et al. Proc. Natl. Acad. Sci. USA 2006 103:11329

2. MV Gammons et al. Invest. Ophthalmol. Vis. Sci. 2013 54:5797

3. MV Gammons et al. Br. J. Cancer 2014 111:477


CAS Registry Number:

218156-96-8


Molecular Formula:

C18H18F3N3O


Appearance:

White powder


Molecular Weight:

349.4


Purity:

>98% (TLC); NMR (Conforms)


Solubilization:

May be dissolved in DMSO (40 mg/ml) or ethanol (25 mg/ml)


Aliases:

N-[2-(1-Piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide


Storage and Stability:

Store desiccated as supplied at -20oC temperature for up to 2 years. Store solutions at -20oC for up to 1 month.


Molecular Structure:



Product Datasheets



There are no related publications available for this product.


RESEARCH AREAS

Cancer, Inflammation, Neurobiology, Ser/Thr Kinases


RELATED PRODUCTS


  SRPK1, Active, S21-10G

  SRPK2, Active, S22-10G


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