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LH-846

Casein Kinase 1δ inhibitor
Catalog No. C67-901


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Catalog No. Pack Size Price (USD)
C67-901-05 5 mg $83
C67-901-25 25 mg $303
C67-901-BULK BULK Contact Us  


Overview:

Selective inhibitor of casein kinase (CK) 1δ, IC50s=0.29, 1.3 and 2.5 µM for δ, ε and α isoforms respectively with no inhibition of CK2. Inhibits CK1δ-mediated phosphorylation.

References:


1. JW Lee et al. Angew. Chem. Int. Ed. Engl. 2011 50:10608


CAS Registry Number:

639052-78-1


Molecular Formula:

C16H13ClN2OS


Appearance:

White crystalline powder


Molecular Weight:

318.81


Purity:

>98% (TLC); NMR (Conforms)


Solubilization:

May be dissolved in DMSO (20 mg/ml) or ethanol (5 mg/ml, warm)


Aliases:

N-(5-Chloro-6-methyl-2-enzothiazolyl)benzeneacetamide


Storage and Stability:

Store desiccated as supplied at ambient temperature for up to 2 years. Store solutions at -20oC for up to 3 months.


Molecular Structure:



Product Datasheets



There are no related publications available for this product.


RELATED PRODUCTS


  Casein Protein, C03-54N

  Casein, Dephosphorylated, C03-54BN


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