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BRD-7389

RSK Inhibitor
Catalog No. R15-901


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Catalog No. Pack Size Price (USD)
R15-901-05 5 mg $105
R15-901-25 25 mg $402
R15-901-BULK BULK Contact Us  


Overview:

Inhibits p90 ribosomal S6 kinase (RSK), IC50 = 1.2, 1.5 and 2.4 µM for RSK3, RSK1 and RSK2 respectively1.

References:


1. D Fomina-Yadlin et al. Proc. Natl. Acad. Sci. USA 2010 107:15099

2. A Choudhary et al. PLoS One 2014 9(4):e95194

3. YS Park and NJ Cho Mol. Cell. Biochem. 2012 370:191


CAS Registry Number:

376382-11-5


Molecular Formula:

C24H18N2O2


Appearance:

Beige Powder


Molecular Weight:

366.41


Purity:

>98% (TLC); NMR (Conforms)


Solubilization:

May be dissolved in DMSO (35 mg/ml)


Aliases:

1-[(2-Phenylethyl)amino]-3H-naphtho[1,2,3-de]quinoline-2,7-dione


Storage and Stability:

Store desiccated as supplied at -20oC for up to 2 years. Store solutions at -20oC for up 3 months.


Molecular Structure:



Product Datasheets



There are no related publications available for this product.


RESEARCH AREAS

Apoptosis/Autophagy, Cancer, Cardiovascular Disease, ERK/MAPK Pathway, Inflammation, Neurobiology, NfkB Pathway, Ser/Thr Kinases


RELATED PRODUCTS


  RSK2 (L608F), Active, R17-12CG

  RSK1, Active, R15-10G

  RSK2, Active, R17-10G

  RSK3, Active, R16-10G


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